Przejdź do zawartości
Merck

EPI003

Sigma-Aldrich

In Situ Histone Deacetylase (HDAC) Activity Fluorometric Assay Kit

100 assays in 96 well plates

Zaloguj sięWyświetlanie cen organizacyjnych i kontraktowych


About This Item

Numer WE:
Kod UNSPSC:
12352200
NACRES:
NA.41

zastosowanie

100 assays in 96 well plates

Warunki transportu

wet ice

temp. przechowywania

−20°C

Opis ogólny

Histone deacetylases (HDACs) are a large family of enzymes that remove acetyl groups from histone proteins. HDACs are localized in both the cytosol and nucleus and some shuttle between the two locations.
Sigma′s InSitu HDAC Activity Fluorometric Assay Kit provides a direct, fast, fluorescence-based method to measure HDAC activity in cultured cells. The procedure requires just two steps, both performed in the original 96-well cell culture plate. First, the cell culture medium is replaced with a cell permeable HDAC Substrate, containing an acetylated lysine side chain. During the subsequent incubation, HDAC Substrate enters the cells and is deacetylated by intracellular HDAC. In the second step, Developer is added to lyse the cells and cleave the deacetylated HDAC Substrate to release a fluorophore. The fluorescence generated can be quantified at Ex/Em = 368/442 nm. The assay is well suited for either individual or high throughput screening.

Zastosowanie

In Situ Histone Deacetylase (HDAC) Activity Fluorometric Assay Kit has been used to determine HDAC activity.

Działania biochem./fizjol.

Site specific histone acetylation and deacetylation have been shown to activate or repress eukaryotic gene transcription, respectively, and as a consequence, histone deacetylases (HDACs) play a crucial role in organism development and disease. Mutation or abnormal expression of HDAC is observed in cancer.

Cechy i korzyści

  • Simple two-step sensitive and reliable assay
  • All steps performed in the same cell culture plate
  • Utilizes fluorometric method
  • Sample type: cultured, adherent, and suspension cells
  • Suitable for individual tests or high throughput assays and kinetic studies
  • Convenient 96-well microplate format
  • Suitable for screening HDAC inhibitors or activators
  • Suitable for studying growth factors or other regulators that influence HDAC activity
Ta strona może zawierać tekst przetłumaczony maszynowo.

Piktogramy

Exclamation mark

Hasło ostrzegawcze

Warning

Zwroty wskazujące rodzaj zagrożenia

Zwroty wskazujące środki ostrożności

Klasyfikacja zagrożeń

Aquatic Chronic 3 - Eye Irrit. 2

Kod klasy składowania

10 - Combustible liquids

Temperatura zapłonu (°F)

188.6 °F - closed cup

Temperatura zapłonu (°C)

87 °C - closed cup


Wybierz jedną z najnowszych wersji:

Certyfikaty analizy (CoA)

Lot/Batch Number

Nie widzisz odpowiedniej wersji?

Jeśli potrzebujesz konkretnej wersji, możesz wyszukać konkretny certyfikat według numeru partii lub serii.

Masz już ten produkt?

Dokumenty związane z niedawno zakupionymi produktami zostały zamieszczone w Bibliotece dokumentów.

Odwiedź Bibliotekę dokumentów

Covalent modifications of histones during development and disease pathogenesis.
Bhaumik S R, et al.
Nature Structural and Molecular Biology, 14(11), 1008-1008 (2007)
The biology of HDAC in cancer: the nuclear and epigenetic components.
Handbook of Experimental Pharmacology, 206, 13-37 (2011)
Targeting histone deacetylase activity to arrest cell growth and promote neural differentiation in Ewing sarcoma.
Souza B K, et al.
Molecular Neurobiology, 1-17 (2018)
Christina Stache et al.
Neurosurgical focus, 41(6), E14-E14 (2016-12-03)
OBJECTIVE In this study, the authors investigated the underlying mechanisms responsible for high tumor recurrence rates of adamantinomatous craniopharyngioma (ACP) after radiotherapy and developed new targeted treatment protocols to minimize recurrence. ACPs are characterized by the activation of the receptor
Long Jin et al.
Theriogenology, 87, 298-305 (2016-10-16)
Cloning remains as an important technique to enhance the reconstitution and distribution of animal population with high-genetic merit. One of the major detrimental factors of this technique is the abnormal epigenetic modifications. MGCD0103 is known as a histone deacetylase inhibitor.

Nasz zespół naukowców ma doświadczenie we wszystkich obszarach badań, w tym w naukach przyrodniczych, materiałoznawstwie, syntezie chemicznej, chromatografii, analityce i wielu innych dziedzinach.

Skontaktuj się z zespołem ds. pomocy technicznej