539636

PKC_θ Pseudosubstrate Inhibitor, Myristoylated

The PKC_θ Pseudosubstrate Inhibitor, Myristoylated controls the biological activity of PKC_θ. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.

• Sinônimo(s): PKC_θ Pseudosubstrate Inhibitor, Myristoylated, Myr-LHQRRGAIKQAKVHHVKC-NH₂, Protein Kinase C _θ Pseudosubstrate Inhibitor, Myristoylated, Myr-LHQRRGAIKQAKVHHVKC-NH₂, Protein Kinase C_θ Pseudosubstrate Inhibitor, Myristoylated
• Fórmula empírica (Notação de Hill): C₁₀₅H₁₈₂N₃₅O₂₂S
• Peso molecular: 2318.85
• Código UNSPSC: 12352200
• NACRES: NA.77

Propriedades

• Nível de qualidade: 100
• Ensaio: ≥95% (HPLC)
• Formulário: lyophilized solid
• fabricante/nome comercial: Calbiochem^®
• condição de armazenamento: OK to freeze; desiccated (hygroscopic)
• solubilidade: water: 2 mg/mL
• Condições de expedição: ambient
• temperatura de armazenamento: −20°C

Descrição

Descrição geral

A cell-permeable, reversible, substrate competitive, myristoylated form of the inhibitor of protein kinase C_θ isozyme pseudosubstrate inhibitor (Cat. No. 539634).

Cell-permeable myristoylated protein kinase Cq pseudosubstrate sequence peptide (Cat. No. 539634). Useful for studies of PKC_θ function in intact cells. Sold on the basis of peptide content.

Ações bioquímicas/fisiológicas

Cell permeable: yes

Primary Target
protein kinase Cθ

Product competes with ATP.

Reversible: yes

Advertência

Toxicity: Standard Handling (A)

Sequência

Myr-Leu-His-Gln-Arg-Arg-Gly-Ala-Ile-Lys-Gln-Ala-Lys-Val-His-His-Val-Lys-Cys-NH₂

forma física

Supplied as a trifluoroacetate salt.

Reconstituição

Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for 6 months at -20°C.

Outras notas

Osada, S., et al. 1992. Mol. Cell Biol.12, 3930.

Informações legais

CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany

Informações de segurança

• Código de classe de armazenamento: 11 - Combustible Solids
• Classe de risco de água (WGK): WGK 1
• Ponto de fulgor (°F): Not applicable
• Ponto de fulgor (°C): Not applicable