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About This Item
經驗公式（希爾表示法）:
C10H16N6S
CAS號碼:
分子量：:
252.34
EC號碼:
MDL號碼:
分類程式碼代碼:
12352200
PubChem物質ID:
NACRES:
NA.77
推薦產品
形狀
powder
起源
GlaxoSmithKline
儲存溫度
2-8°C
SMILES 字串
CN\C(NC#N)=N\CCSCc1nc[nH]c1C
InChI
1S/C10H16N6S/c1-8-9(16-7-15-8)5-17-4-3-13-10(12-2)14-6-11/h7H,3-5H2,1-2H3,(H,15,16)(H2,12,13,14)
InChI 密鑰
AQIXAKUUQRKLND-UHFFFAOYSA-N
基因資訊
human ... ABCB1(5243) , CYP1A2(1544) , CYP3A4(1576) , HRH2(3274) , SLC9A2(6549) , SLC9A5(6553)
mouse ... Abcb1a(18671) , Abcb1b(18669)
rat ... Slc9a1(24782) , Slc9a3(24784) , Slc9a5(192215)
尋找類似的產品？ 前往 產品比較指南
生化／生理作用
H2组胺受体拮抗剂；I1咪唑啉受体激动剂；抗溃疡剂。通过抑制内皮细胞表面上E-选择蛋白的表达来阻断癌症转移，从而阻断肿瘤细胞的粘附。
特點和優勢
该化合物由 GlaxoSmithKline 开发。想要浏览其他由制药公司开发的化合物以及已批准药物/候选药物清单，请单击此处。
这种化合物是 ADME 毒性研究的特色产品。点击此处发现更多特色 ADME 毒性产品。在sigma.com/discover-bsm可了解更多关于生物活性小分子的其他研究领域。
儲存類別代碼
11 - Combustible Solids
水污染物質分類（WGK）
WGK 3
個人防護裝備
Eyeshields, Gloves, type P3 (EN 143) respirator cartridges
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