539604

PKC_η Pseudosubstrate Inhibitor, Myristoylated

The PKC_η Pseudosubstrate Inhibitor, Myristoylated controls the biological activity of PKC_η. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.

• Synonym(e): PKC_η Pseudosubstrate Inhibitor, Myristoylated, Myr-TRKRQRAMRRRVHQING-OH, Protein Kinase C _η Pseudosubstrate Inhibitor, Myristoylated
• Empirische Formel (Hill-System): C₁₀₁H₁₈₅N₄₁O₂₃S
• Molekulargewicht: 2373.88
• UNSPSC-Code: 12352200
• NACRES: NA.77

Eigenschaften

• Qualitätsniveau: 100
• Assay: ≥95% (HPLC)
• Form: lyophilized solid
• Hersteller/Markenname: Calbiochem^®
• Lagerbedingungen: OK to freeze; desiccated (hygroscopic)
• Löslichkeit: water: 1 mg/mL
• Versandbedingung: ambient
• Lagertemp.: −20°C

Beschreibung

Allgemeine Beschreibung

A cell-permeable, reversible, substrate competitive, and pseudosubstrate inhibitor of the protein kinase C_η isozyme. Useful for studies of PKC_η function in intact cells.

Biochem./physiol. Wirkung

Cell permeable: yes

Primary Target
PKCν

Product competes with ATP.

Reversible: yes

Verpackung

Yes

Warnhinweis

Toxicity: Standard Handling (A)

Sequenz

Myr-Thr-Arg-Lys-Arg-Gln-Arg-Ala-Met-Arg-Arg-Arg-Val-His-Gln-Ile-Asn-Gly-OH

Physikalische Form

Supplied as a trifluoroacetate salt.

Rekonstituierung

Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 6 months at -20°C.

Sonstige Hinweise

Osada, S., et al. 1992. Mol. Cell Biol.12, 3930.

Rechtliche Hinweise

CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany

Sicherheitshinweise

• Lagerklassenschlüssel: 11 - Combustible Solids
• WGK: WGK 1
• Flammpunkt (°F): Not applicable
• Flammpunkt (°C): Not applicable