Pular para o conteúdo
Merck
Todas as fotos(2)

Documentos Principais

SRP5089

Sigma-Aldrich

TBK1, active, GST tagged human

PRECISIO® Kinase, recombinant, expressed in baculovirus infected Sf9 cells, ≥70% (SDS-PAGE), buffered aqueous glycerol solution

Sinônimo(s):

FLJ11330, NAK, T2K

Faça loginpara ver os preços organizacionais e de contrato


About This Item

Código UNSPSC:
12352204
NACRES:
NA.32

recombinante

expressed in baculovirus infected Sf9 cells

linha de produto

PRECISIO® Kinase

Ensaio

≥70% (SDS-PAGE)

Formulário

buffered aqueous glycerol solution

atividade específica

259-351 nmol/min·mg

peso molecular

~105 kDa

nº de adesão NCBI

Condições de expedição

dry ice

temperatura de armazenamento

−70°C

Informações sobre genes

human ... TBK1(29110)

Descrição geral

TBK1 (TANK-binding kinase 1) gene is located on human chromosome 12q14. It is a serine/threonine protein kinase. The encoded protein has a kinase domain, a ubiquitin-like domain, an α-helical scaffold dimerization domain and a small adaptor-binding motif.

Ações bioquímicas/fisiológicas

TBK1 (TANK-binding kinase 1) can phosphorylate numerous proteins, like optineurin, P62 (sequestosome 1) and interferon regulatory factor 3 (IRF3). It participates in various signaling pathways, namely, autophagy, antiviral and antibacterial innate immunity responses, oncogenic transformation and expression of inflammatory mediators. Mutations in this gene are linked with sporadic amyotrophic lateral sclerosis (SALS), familial ALS (FALS) and frontotemporal dementia. Defects in TBK1 suppresses autophagy, causing the accumulation of damaged mitochondria, thereby leading to neurodegeneration. Alteration in the copy number of TBK1 gene is associated with normal tension glaucoma. TBK1, also known as NAK or NFκB-activating kinase, is an upstream protein kinase that can phosphorylate and activate the IkB kinases. Activation of IkB kinases allows the phosphorylation of IkB protein which is then degraded via the ubiquitination pathway. This mechanism allows the activation of the NFκB transcriptional complex. TBK1 is a specific upstream regulator of IkB kinases and can also interact and the IkB protein TANK. TBK1 is a component of the virus-activated kinase that phosphorylate IRF3 and IRF7 allowing their dimerization and translocation to the nucleus, where they induce transcription of interferon.

forma física

Supplied in 50mM Tris-HCl, pH 7.5, 150mM NaCl, 10mM glutathione, 0.1mM EDTA, 0.25mM DTT, 0.1mM PMSF, 25% glycerol.

Nota de preparo

after opening, aliquot into smaller quantities and store at -70 °C. Avoid repeating handling and multiple freeze/thaw cycles

Informações legais

PRECISIO is a registered trademark of Merck KGaA, Darmstadt, Germany

Código de classe de armazenamento

10 - Combustible liquids

Classe de risco de água (WGK)

WGK 1


Escolha uma das versões mais recentes:

Certificados de análise (COA)

Lot/Batch Number

Não está vendo a versão correta?

Se precisar de uma versão específica, você pode procurar um certificado específico pelo número do lote ou da remessa.

Já possui este produto?

Encontre a documentação dos produtos que você adquiriu recentemente na biblioteca de documentos.

Visite a Biblioteca de Documentos

Confirmation of TBK1 duplication in normal tension glaucoma
Kawase K, et al.
Experimental Eye Research, 96(1), 178-178 (2012)
Mutational analysis of TBK1 in Taiwanese patients with amyotrophic lateral sclerosis
Tsai PC , et al.
Neurobiology of Aging, 40, 191-e11-191-e11 (2016)
Dynamic recruitment and activation of ALS-associated TBK1 with its target optineurin are required for efficient mitophagy
Moore AS and Holzbaur ELF
Proceedings of the National Academy of Sciences of the USA, 113(24), E3349-E3358 (2016)
Loss of TBK1 is a frequent cause of frontotemporal dementia in a Belgian cohort
Gijselinck I, et al.
Neurology, 85(24), 2116-2125 (2015)
Y Tojima et al.
Nature, 404(6779), 778-782 (2000-04-28)
Phosphorylation of IkappaB by the IkappaB kinase (IKK) complex is a critical step leading to IkappaB degradation and activation of transcription factor NF-kappaB. The IKK complex contains two catalytic subunits, IKKalpha and IKKbeta, the latter being indispensable for NF-kappaB activation

Nossa equipe de cientistas tem experiência em todas as áreas de pesquisa, incluindo Life Sciences, ciência de materiais, síntese química, cromatografia, química analítica e muitas outras.

Entre em contato com a assistência técnica