R1908

Remifentanil hydrochloride

≥97% (HPLC), powder

• 別名: 3-[methoxycarbonyl-4-[(1-oxopropyl)phenylamino]1-piperidine]propanoic acid methyl ester hydrochloride, GI-87084B, Remifentanyl, Ultiva
• 実験式（ヒル表記法）: C₂₀H₂₈N₂O₅·HCl
• CAS番号: 132539-07-2
• 分子量: 412.91
• MDL番号: MFCD00910882
• UNSPSCコード: 12352200
• PubChem Substance ID: 329824010

特性

• 品質水準: 100
• アッセイ: ≥97% (HPLC)
• フォーム: powder
• 薬剤管理: USDEA Schedule II; regulated under CDSA - not available from Sigma-Aldrich Canada; estupefaciente (Spain); Decreto Lei 15/93: Tabela IA (Portugal)
• 保管条件: desiccated
• 色: white to off-white
• 溶解性: H₂O: ≥20 mg/mL
• 保管温度: 2-8°C
• SMILES記法: O=C(CC)N(C1(CCN(CCC(OC)=O)CC1)C(OC)=O)C2=CC=CC=C2.[H]Cl
• InChI: 1S/C20H28N2O5.ClH/c1-4-17(23)22(16-8-6-5-7-9-16)20(19(25)27-3)11-14-21(15-12-20)13-10-18(24)26-2;/h5-9H,4,10-15H2,1-3H3;1H
• InChI Key: WFBMIPUMYUHANP-UHFFFAOYSA-N
• 遺伝子情報: human ... OPRM1(4988)

詳細

生物化学的／生理学的作用

Remifentanil hydrochloride is a mu opioid receptor agonist, anesthetic, and analgesic compound. Remifentanil was developed as an ultra-short-acting mu opioid receptor agonist with improved pharmacodynamic properties.

特徴および利点

This compound is featured on the Opioid Receptors page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.

安全性情報

• ピクトグラム: GHS08
• シグナルワード: Warning
• 危険有害性情報: H371
• 注意書き: P260 - P264 - P270 - P308 + P311 - P405 - P501
• 危険有害性の分類: STOT SE 2
• ターゲットの組織: Respiratory system
• 保管分類コード: 11 - Combustible Solids
• WGK: WGK 1
• 引火点(°F): Not applicable
• 引火点(℃): Not applicable