推薦產品
品質等級
化驗
>97%
形狀
solid
顏色
white
溶解度
H2O: 89 mg/mL
SMILES 字串
O[C@H]([C@@H](O)C(O)=O)C(O)=O.CCN1CCC[C@H]1CNC(=O)c2c(O)c(Cl)cc(Cl)c2OC
InChI
1S/C15H20Cl2N2O3.C4H6O6/c1-3-19-6-4-5-9(19)8-18-15(21)12-13(20)10(16)7-11(17)14(12)22-2;5-1(3(7)8)2(6)4(9)10/h7,9,20H,3-6,8H2,1-2H3,(H,18,21);1-2,5-6H,(H,7,8)(H,9,10)/t9-;1-,2-/m01/s1
InChI 密鑰
QULBVRZTKPQGCR-NDAAPVSOSA-N
基因資訊
human ... DRD2(1813)
應用
S(−)-雷氯必利(+)-酒石酸盐已用作D2 受体拮抗剂:
- 研究D2受体在介导动物PAG腹外侧区(vlPAG)/背侧中缝多巴胺能镇痛中的作用
- Thap1缺失小鼠药理学和行为研究
- 测定Ca2+瞬变与大鼠多巴胺神经元活性之间的关系
生化/生理作用
雷氯必利是一种苯甲酰胺衍生物和选择性D2多巴胺受体拮抗剂。
包裝
无底玻璃瓶。内含物装在插入的融合锥内。
注意
光敏性
儲存類別代碼
11 - Combustible Solids
水污染物質分類(WGK)
WGK 3
閃點(°F)
Not applicable
閃點(°C)
Not applicable
個人防護裝備
Eyeshields, Gloves, type N95 (US)
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