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About This Item
經驗公式（希爾表示法）:
C25H30N6O2 · 2HCl
CAS號碼:
分子量：:
519.47
MDL號碼:
分類程式碼代碼:
12352204
PubChem物質ID:
NACRES:
NA.32
推薦產品
產品名稱
苯丙氨酸-精氨酸 β-萘胺 二盐酸盐, cathepsin substrate
品質等級
化驗
≥98% (TLC)
形狀
powder
溶解度
water: 50 mg/mL, clear, colorless to faintly yellow
儲存溫度
−20°C
SMILES 字串
Cl.NC(Cc1ccccc1)C(=O)NC(CCCNC(N)=N)C(=O)Nc2ccc3ccccc3c2
InChI
1S/C25H30N6O2.ClH/c26-21(15-17-7-2-1-3-8-17)23(32)31-22(11-6-14-29-25(27)28)24(33)30-20-13-12-18-9-4-5-10-19(18)16-20;/h1-5,7-10,12-13,16,21-22H,6,11,14-15,26H2,(H,30,33)(H,31,32)(H4,27,28,29);1H
InChI 密鑰
ZMTAZQYLEGNUTJ-UHFFFAOYSA-N
一般說明
Phe-Arg β-萘酰胺，一种拟肽化合物， 是一种外排泵抑制剂（EPI）。它可作用于革兰氏阴性细菌的主要多药耐药性外向转运蛋白。Phe-Arg-萘酰胺可在铜绿假单胞菌中降低氟喹诺酮类药物的耐药性。
應用
Phe-Arg-萘酰胺二盐酸盐用于评估外排泵对抗菌素耐药性的贡献。在存在外排泵抑制剂的条件下，它还用于最小抑菌浓度测试。
包裝
无底玻璃瓶。内含物在插入的融合锥体内。
基底
二肽基氨肽酶I（组织蛋白酶C）的底物。
儲存類別代碼
11 - Combustible Solids
水污染物質分類（WGK）
WGK 3
閃點（°F）
Not applicable
閃點（°C）
Not applicable
個人防護裝備
Eyeshields, Gloves, type N95 (US)
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