539610

PKC_ζ/ι Pseudosubstrate Inhibitor

The PKC_ζ/ι Pseudosubstrate Inhibitor controls the biological activity of PKC_ζ/ι. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.

• 同義詞: PKC_ζ/ι Pseudosubstrate Inhibitor, SIYRRGARRWRKL, Protein Kinase C _ζ/ι Pseudosubstrate Inhibitor, SIYRRGARRWRKL, Protein Kinase C_ζ/ι Pseudosubstrate Inhibitor
• 經驗公式（希爾表示法）: C₇₆H₁₂₈N₃₀O₁₆
• 分子量：: 1718.02
• 分類程式碼代碼: 12352200
• NACRES: NA.77

屬性

• 品質等級: 100
• 化驗: ≥95% (HPLC)
• 形狀: lyophilized
• 製造商／商標名: Calbiochem^®
• 儲存條件: OK to freeze; desiccated (hygroscopic)
• 溶解度: glacial acetic acid: 2 mg/mL; water: 2 mg/mL
• 運輸包裝: ambient
• 儲存溫度: −20°C

描述

一般說明

A selective, reversible, and substrate competitive inhibitor of protein kinase C_ζ and protein kinase C_ι (PKC_ζ/ι) isozymes.

Non-cell-permeable protein kinase C_ζ and protein kinase C_ι pseudosubstrate sequence peptide that can be used as a selective, reversible, and substrate competitive inhibitor PKC_ζ/ι in in vitro kinase assays.

生化／生理作用

Cell permeable: no

Primary Target
PKCζ

Product does not compete with ATP.

Reversible: yes

警告

Toxicity: Standard Handling (A)

序列

H-Ser-Ile-Tyr-Arg-Arg-Gly-Ala-Arg-Arg-Trp-Arg-Lys-Leu-OH

外觀

Supplied as a trifluoroacetate salt.

重構

Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.

其他說明

Sajan, M.P., et al. 1999. J. Biol. Chem.274, 30495.
Laudanna, C., et al. 1998. J. Biol. Chem.273, 30306.
Standaert, M.L., et al. 1997. J. Biol. Chem.272, 30075.

法律資訊

CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany

安全資訊

• 儲存類別代碼: 11 - Combustible Solids
• 水污染物質分類（WGK）: WGK 1
• 閃點（°F）: Not applicable
• 閃點（°C）: Not applicable