推薦產品
品質等級
化驗
≥95.0%
形狀
solid
mp
>300 °C (lit.)
SMILES 字串
OB(O)c1cccnc1
InChI
1S/C5H6BNO2/c8-6(9)5-2-1-3-7-4-5/h1-4,8-9H
InChI 密鑰
ABMYEXAYWZJVOV-UHFFFAOYSA-N
應用
3-吡啶基硼酸可用作以下反应中的试剂:
它也可用于制备:
- 不含磷的Suzuki-Miyaura交叉偶联反应
- 区域选择性Suzuki-Miyaura偶联和串联钯催化的分子内氨基羰基化和环化
- 乙酰丙酮铜催化的N-芳基化反应
- 铜介导的富电子苯的氰化和区域选择性氰化反应
它也可用于制备:
- 通过Suzuki偶联反应制备新型线性聚(苯基吡啶基)链
- 低聚吡啶基折叠体,作为α-螺旋扭曲结构的模拟物
- 许多非常重要的治疗性酶和激酶抑制剂以及受体拮抗剂
- 通过Suzuki偶联反应与二溴吡啶胺化物反应生成吡啶取代的吡啶N-(2′-叠氮基)胺化物。
其他說明
含不定量的酸酐
儲存類別代碼
11 - Combustible Solids
水污染物質分類(WGK)
WGK 3
閃點(°F)
Not applicable
閃點(°C)
Not applicable
個人防護裝備
Eyeshields, Gloves, type N95 (US)
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文章
This brochure contains a comprehensive selection of boronic acids, boronic acid esters, diboron esters, and transition-metal catalysts useful for the Suzuki–Miyaura coupling reaction
This brochure contains a comprehensive selection of boronic acids, boronic acid esters, diboron esters, and transition-metal catalysts useful for the Suzuki–Miyaura coupling reaction
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