5.08160

DPDPE

• 别名: DPDPE, δ Opioid Receptor Agonist, DPDPE
• 经验公式（希尔记法）: C₃₀H₃₉N₅O₇S₂
• CAS号: 88373-73-3
• 分子量: 645.79
• 分類程式碼代碼: 12352200
• NACRES: NA.77

属性

• 化驗: ≥99% (HPLC)
• 品質等級: 100
• 形狀: solid
• 製造商／商標名: Calbiochem^®
• 儲存條件: OK to freeze; protect from light
• 顏色: off-white
• 溶解度: water: 1 mg/mL
• 儲存溫度: −20°C
• InChI: 1S/C30H39N5O7S2/c1-29(2)23(34-25(38)20(31)14-18-10-12-19(36)13-11-18)27(40)32-16-22(37)33-21(15-17-8-6-5-7-9-17)26(39)35-24(28(41)42)30(3,4)44-43-29/h5-13,20-21,23-24,36H,14-16,31H2,1-4H3,(H,32,40)(H,33,37)(H,34,38)(H,35,39)(H,41,42)/t20-,21-,23-,24-/m0/s1
• InChI 密鑰: MCMMCRYPQBNCPH-WMIMKTLMSA-N

说明

一般說明

A potent agonist selective for δ opioid receptor (EC₅₀ = 5.2 nM). Exhibits anti-convulsant effects in vivo in rats, also used in nociceptive studies.

生化／生理作用

Primary Target
δ opioid receptor

警告

Toxicity: Standard Handling (A)

序列

Tyr-D-Pen-Gly-Phe-D-Pen (2-5 disulfide bond)

重構

Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.

其他說明

Chen, C., 1997. J. Pharmacol. Exp. Ther.283, 1151.
Chandrakumar, S., et al., 1992. J. Med. Chem.35, 2928.
Tortella, F. 1988. Peptides.9, 1177.
Clark, A., et al., 1986. Eur. J. Pharmacol.128, 303.

法律資訊

CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany

安全信息

• 儲存類別代碼: 11 - Combustible Solids
• 水污染物質分類（WGK）: WGK 3
• 閃點（°F）: Not applicable
• 閃點（°C）: Not applicable