924229

(S,R,S)-AHPC-Me

95%

• Sinônimo(s): (2S,4R)-1-((S)-2-amino-3,3-dimethylbutanoyl)-4-hydroxy-N-((S)-1-(4-(4-methylthiazol-5-yl)phenyl)ethyl)pyrrolidine-2-carboxamide, PROTAC^® research ligand, VH032 methyl derivative
• Fórmula empírica (Notação de Hill): C₂₃H₃₂N₄O₃S
• Número CAS: 1948273-02-6
• Peso molecular: 444.59
• Número MDL: MFCD31630815
• Código UNSPSC: 12352101
• NACRES: NA.22

Propriedades

• ligand: VH032
• Nível de qualidade: 100
• Ensaio: 95%
• forma: powder
• temperatura de armazenamento: 2-8°C
• cadeia de caracteres SMILES: C([C@H](C(C)(C)C)N)(=O)N1[C@H](C(N[C@@H](C)C2=CC=C(C=C2)C3=C(C)N=CS3)=O)C[C@@H](O)C1

Descrição

Aplicação

(S,R,S)-AHPC-Me is a VH032 derivative used in the recruitment of the von Hippel-Lindau (VHL) protein for targeted protein degradation and PROTAC (proteolysis-targeting chimeras) technology. This was previously listed under ATEH961B8E6E.

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Informações legais

PROTAC is a registered trademark of Arvinas Operations, Inc., and is used under license

Informações de segurança

• Código de classe de armazenamento: 11 - Combustible Solids
• Classe de risco de água (WGK): WGK 3
• Ponto de fulgor (°F): Not applicable
• Ponto de fulgor (°C): Not applicable