推薦產品
品質等級
化驗
≥90% (HPLC)
形狀
powder
儲存條件
desiccated
顏色
white to beige
溶解度
DMSO: >5 mg/mL
儲存溫度
2-8°C
SMILES 字串
COc1ccc(cc1)C(=O)c2c(C)n(CCN3CCOCC3)c4cc(I)ccc24
InChI
1S/C23H25IN2O3/c1-16-22(23(27)17-3-6-19(28-2)7-4-17)20-8-5-18(24)15-21(20)26(16)10-9-25-11-13-29-14-12-25/h3-8,15H,9-14H2,1-2H3
InChI 密鑰
JHOTYHDSLIUKCJ-UHFFFAOYSA-N
應用
AM630 已被用于：
- 作为大麻素2（CB2）抑制剂用于研究变色栓菌多糖肽 (TPSP) 的镇痛作用。
- 作为CB2拮抗剂与β-石竹烯（BCP）一起用于研究其对成纤维细胞再上皮化的作用。
- 作为CB2拮抗剂用于研究其与原代人成骨细胞中的17-β-雌二醇的相互作用。
生化／生理作用
AM630 是一种选择性 CB2 大麻素拮抗剂/反向激动剂（Ki = 31.2 nM），选择性比CB1 受体大150倍。
AM630是一种氨基烷基吲哚，可作为CP 55,940和WIN 55,212-2的竞争性拮抗剂。它也可作为大麻素和（R）-（+）-花生四烯基-1′-羟基-2′-丙酰胺（AM356）的竞争性拮抗剂。
訊號詞
Warning
危險聲明
危險分類
Aquatic Acute 1 - Aquatic Chronic 1
儲存類別代碼
11 - Combustible Solids
水污染物質分類（WGK）
WGK 3
閃點（°F）
Not applicable
閃點（°C）
Not applicable
分析證明 (COA)
輸入產品批次/批號來搜索 分析證明 (COA)。在產品’s標籤上找到批次和批號，寫有 ‘Lot’或‘Batch’.。
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