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Merck

R134

Sigma-Aldrich

Rilmenidine hemifumarate salt

solid

别名:

N-(Dicyclopropylmethyl)-4,5-dihydro-2-oxazolamine hemifumarate salt, Oxaminozoline hemifumarate salt, Rilmenidene hemifumarate salt

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About This Item

经验公式(希尔记法):
C10H16N2O · 0.5C4H4O4
分子量:
238.28
MDL號碼:
分類程式碼代碼:
12352200
PubChem物質ID:
NACRES:
NA.77

形狀

solid

顏色

white

溶解度

DMSO: >10 mg/mL
H2O: insoluble

起源

Servier

SMILES 字串

OC(=O)\C=C\C(O)=O.C1CN=C(NC(C2CC2)C3CC3)O1.C4CN=C(NC(C5CC5)C6CC6)O4

InChI

1S/2C10H16N2O.C4H4O4/c2*1-2-7(1)9(8-3-4-8)12-10-11-5-6-13-10;5-3(6)1-2-4(7)8/h2*7-9H,1-6H2,(H,11,12);1-2H,(H,5,6)(H,7,8)/b;;2-1+

InChI 密鑰

LZFATBMLSYHRTC-WXXKFALUSA-N

基因資訊

human ... NISCH(11188)

生化/生理作用

Selective I1 imidazoline receptor agonist.

特點和優勢

This compound is featured on the Imidazoline Binding Sites page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.
This compound was developed by Servier. To browse the list of other pharma-developed compounds and Approved Drugs/Drug Candidates, click here.

儲存類別代碼

11 - Combustible Solids

水污染物質分類(WGK)

WGK 3

閃點(°F)

Not applicable

閃點(°C)

Not applicable

個人防護裝備

Eyeshields, Gloves, type N95 (US)


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K Takada et al.
British journal of pharmacology, 120(8), 1575-1581 (1997-04-01)
1. To elucidate the possible involvement of pertussis toxin (PTX)-sensitive G proteins in the post receptor mechanism of alpha 2-adrenoceptors and imidazoline receptors, we examined the effect of pretreatment of the central nervous system with PTX on the antidysrhythmic effect
C K Chan et al.
The Journal of pharmacology and experimental therapeutics, 276(2), 411-420 (1996-02-01)
The present study in conscious rabbits with intracisternal (i.c.) catheters sought to determine the relative contribution of the I1 subtype of imidazoline receptors (IR) and alpha 2 adrenoceptors to the hypotensive effects of rilmenidine, clonidine and moxonidine with an I1-IR/alpha
M A Ozog et al.
Journal of neurochemistry, 71(4), 1429-1435 (1998-09-29)
Rilmenidine, a ligand for imidazoline and alpha2-adrenergic receptors, is neuroprotective following focal cerebral ischemia. We investigated the effects of rilmenidine on cytosolic free Ca2+ concentration ([Ca2+]i) in rat astrocytes. Rilmenidine caused concentration-dependent elevation of [Ca2+]i, consisting of a transient increase

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