R134
Rilmenidine hemifumarate salt
solid
동의어(들):
N-(Dicyclopropylmethyl)-4,5-dihydro-2-oxazolamine hemifumarate salt, Oxaminozoline hemifumarate salt, Rilmenidene hemifumarate salt
로그인조직 및 계약 가격 보기
모든 사진(2)
About This Item
실험식(Hill 표기법):
C10H16N2O · 0.5C4H4O4
CAS Number:
Molecular Weight:
238.28
MDL number:
UNSPSC 코드:
12352200
PubChem Substance ID:
NACRES:
NA.77
추천 제품
양식
solid
색상
white
solubility
DMSO: >10 mg/mL
H2O: insoluble
주관자
Servier
SMILES string
OC(=O)\C=C\C(O)=O.C1CN=C(NC(C2CC2)C3CC3)O1.C4CN=C(NC(C5CC5)C6CC6)O4
InChI
1S/2C10H16N2O.C4H4O4/c2*1-2-7(1)9(8-3-4-8)12-10-11-5-6-13-10;5-3(6)1-2-4(7)8/h2*7-9H,1-6H2,(H,11,12);1-2H,(H,5,6)(H,7,8)/b;;2-1+
InChI key
LZFATBMLSYHRTC-WXXKFALUSA-N
유전자 정보
human ... NISCH(11188)
관련 카테고리
생화학적/생리학적 작용
Selective I1 imidazoline receptor agonist.
특징 및 장점
This compound is featured on the Imidazoline Binding Sites page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.
This compound was developed by Servier. To browse the list of other pharma-developed compounds and Approved Drugs/Drug Candidates, click here.
Storage Class Code
11 - Combustible Solids
WGK
WGK 3
Flash Point (°F)
Not applicable
Flash Point (°C)
Not applicable
개인 보호 장비
Eyeshields, Gloves, type N95 (US)
가장 최신 버전 중 하나를 선택하세요:
K Takada et al.
British journal of pharmacology, 120(8), 1575-1581 (1997-04-01)
1. To elucidate the possible involvement of pertussis toxin (PTX)-sensitive G proteins in the post receptor mechanism of alpha 2-adrenoceptors and imidazoline receptors, we examined the effect of pretreatment of the central nervous system with PTX on the antidysrhythmic effect
C K Chan et al.
The Journal of pharmacology and experimental therapeutics, 276(2), 411-420 (1996-02-01)
The present study in conscious rabbits with intracisternal (i.c.) catheters sought to determine the relative contribution of the I1 subtype of imidazoline receptors (IR) and alpha 2 adrenoceptors to the hypotensive effects of rilmenidine, clonidine and moxonidine with an I1-IR/alpha
M A Ozog et al.
Journal of neurochemistry, 71(4), 1429-1435 (1998-09-29)
Rilmenidine, a ligand for imidazoline and alpha2-adrenergic receptors, is neuroprotective following focal cerebral ischemia. We investigated the effects of rilmenidine on cytosolic free Ca2+ concentration ([Ca2+]i) in rat astrocytes. Rilmenidine caused concentration-dependent elevation of [Ca2+]i, consisting of a transient increase
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