539636

PKC_θ Pseudosubstrate Inhibitor, Myristoylated

The PKC_θ Pseudosubstrate Inhibitor, Myristoylated controls the biological activity of PKC_θ. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.

• Synonym(e): PKC_θ Pseudosubstrate Inhibitor, Myristoylated, Myr-LHQRRGAIKQAKVHHVKC-NH₂, Protein Kinase C _θ Pseudosubstrate Inhibitor, Myristoylated, Myr-LHQRRGAIKQAKVHHVKC-NH₂, Protein Kinase C_θ Pseudosubstrate Inhibitor, Myristoylated
• Empirische Formel (Hill-System): C₁₀₅H₁₈₂N₃₅O₂₂S
• Molekulargewicht: 2318.85
• UNSPSC-Code: 12352200
• NACRES: NA.77

Eigenschaften

• Qualitätsniveau: 100
• Assay: ≥95% (HPLC)
• Form: lyophilized solid
• Hersteller/Markenname: Calbiochem^®
• Lagerbedingungen: OK to freeze; desiccated (hygroscopic)
• Löslichkeit: water: 2 mg/mL
• Versandbedingung: ambient
• Lagertemp.: −20°C

Beschreibung

Allgemeine Beschreibung

A cell-permeable, reversible, substrate competitive, myristoylated form of the inhibitor of protein kinase C_θ isozyme pseudosubstrate inhibitor (Cat. No. 539634).

Cell-permeable myristoylated protein kinase Cq pseudosubstrate sequence peptide (Cat. No. 539634). Useful for studies of PKC_θ function in intact cells. Sold on the basis of peptide content.

Biochem./physiol. Wirkung

Cell permeable: yes

Primary Target
protein kinase Cθ

Product competes with ATP.

Reversible: yes

Warnhinweis

Toxicity: Standard Handling (A)

Sequenz

Myr-Leu-His-Gln-Arg-Arg-Gly-Ala-Ile-Lys-Gln-Ala-Lys-Val-His-His-Val-Lys-Cys-NH₂

Physikalische Form

Supplied as a trifluoroacetate salt.

Rekonstituierung

Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for 6 months at -20°C.

Sonstige Hinweise

Osada, S., et al. 1992. Mol. Cell Biol.12, 3930.

Rechtliche Hinweise

CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany

Sicherheitshinweise

• Lagerklassenschlüssel: 11 - Combustible Solids
• WGK: WGK 1
• Flammpunkt (°F): Not applicable
• Flammpunkt (°C): Not applicable