UC168

(±)-Bufuralol hydrochloride

≥98% (HPLC), solid, β-Adrenoceptor agonist/antagonist

• Synonym(e): α-[(tert-Butylamino)methyl]-7-ethyl-2-benzofuranmethanol hydrochloride
• Empirische Formel (Hill-System): C₁₆H₂₃NO₂·HCl
• CAS-Nummer: 60398-91-6
• Molekulargewicht: 297.82
• EG-Nummer: 262-216-3
• MDL-Nummer: MFCD00272648
• UNSPSC-Code: 12161501
• PubChem Substanz-ID: 24724644
• NACRES: NA.77

Eigenschaften

• Produktbezeichnung: (±)-Bufuralol hydrochloride,
• Form: solid
• Qualitätsniveau: 200
• Farbe: white to off-white
• mp (Schmelzpunkt): 143-146 °C
• Löslichkeit: H₂O: soluble; methanol: soluble
• Lagertemp.: 2-8°C
• SMILES String: Cl.CCc1cccc2cc(oc12)C(O)CNC(C)(C)C
• InChI: 1S/C16H23NO2.ClH/c1-5-11-7-6-8-12-9-14(19-15(11)12)13(18)10-17-16(2,3)4;/h6-9,13,17-18H,5,10H2,1-4H3;1H
• InChIKey: KJBONRGCLLBWCJ-UHFFFAOYSA-N

Beschreibung

Anwendung

CYP2D6 substrate

Biochem./physiol. Wirkung

Bufuralol hydrochloride is known to be a non-specific β-receptor inhibitor that has an affinity for β 1 and β 2 receptors. Furthermore, studies have reported that bufuralol hydrochloride can decrease isoproterenol peripheral resistance.

β-Blocker. Varying β-adrenoceptor agonist/antagonist activity.

Leistungsmerkmale und Vorteile

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Verpackung

Bottomless glass bottle. Contents are inside inserted fused cone.

Angaben zur Herstellung

(±)-Bufuralol hydrochloride is soluble in water and methanol.

Sicherheitshinweise

• Lagerklassenschlüssel: 11 - Combustible Solids
• WGK: WGK 3
• Flammpunkt (°F): Not applicable
• Flammpunkt (°C): Not applicable
• Persönliche Schutzausrüstung: dust mask type N95 (US), Eyeshields, Gloves