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Merck

CHRM1

cholinergic receptor, muscarinic 1

Sinonimi:
HM1, M1, M1R
Specie:
ID UniProtKB:
ID gene:
  • Human(1128) Summary: The muscarinic cholinergic receptors belong to a larger family of G protein-coupled receptors. The functional diversity of these receptors is defined by the binding of acetylcholine and includes cellular responses such as adenylate cyclase inhibition, phosphoinositide degeneration, and potassium channel mediation. Muscarinic receptors influence many effects of acetylcholine in the central and peripheral nervous system. The muscarinic cholinergic receptor 1 is involved in mediation of vagally-induced bronchoconstriction and in the acid secretion of the gastrointestinal tract. The gene encoding this receptor is localized to 11q13. [provided by RefSeq, Jul 2008]
  • Mouse(12669) cholinergic receptor, muscarinic 1, CNS
  • Rat(25229) cholinergic receptor, muscarinic 1
  • cow(281684) cholinergic receptor, muscarinic 1
  • Horse(100064117) cholinergic receptor, muscarinic 1
  • domestic cat(101093801) cholinergic receptor, muscarinic 1
  • domestic cat(493664) cholinergic receptor, muscarinic 1
  • dog(483776) cholinergic receptor, muscarinic 1
  • naked mole-rat(101702102) cholinergic receptor, muscarinic 1
  • domestic guinea pig(100728041) cholinergic receptor, muscarinic 1
  • sheep(101117029) cholinergic receptor, muscarinic 1

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Small Molecule - Agonist

Product Number
Descrizione
Specie
Pilocarpine Hydrochloride, Pharmaceutical Secondary Standard; Certified Reference Material,
Specie
human
Pilocarpine hydrochloride, United States Pharmacopeia (USP) Reference Standard,
Specie
human
Pilocarpine nitrate, United States Pharmacopeia (USP) Reference Standard,
Specie
human
Pilocarpine hydrochloride, phyproof® Reference Substance,
Specie
human
Pilocarpine hydrochloride, European Pharmacopoeia (EP) Reference Standard,
Specie
human

Small Molecule - Antagonist

Product Number
Descrizione
Specie
Quinuclidine, 97%,
Specie
rat
Ethopropazine hydrochloride, ≥98% (HPLC), powder,
Specie
human
Scopolamine Hydrobromide, Pharmaceutical Secondary Standard; Certified Reference Material,
Specie
human
Benztropine mesylate, ≥98% (HPLC),
Specie
human
Pirenzepine dihydrochloride, ≥98% (TLC), powder,
Specie
human

Antibodies

Product Number
Descrizione
Reattività con
Applicazione
Anti-Muscarinic Acetylcholine Receptor m1 Antibody, Chemicon®, from rabbit,
Reattività con
mouse, rat
Applicazione
immunohistochemistry
western blot
Anti-CHRM1 antibody produced in rabbit, Prestige Antibodies® Powered by Atlas Antibodies, affinity isolated antibody, buffered aqueous glycerol solution,
Reattività con
human
Applicazione
immunohistochemistry
Anti-CHRM1 antibody produced in rabbit, affinity isolated antibody,
Reattività con
human, mouse, rat
Applicazione
ELISA
western blot
Anti-Muscarinic Acetylcholine Receptor (M1) antibody produced in rabbit, affinity isolated antibody, lyophilized powder,
Reattività con
mouse, rat
Applicazione
immunohistochemistry
western blot

Small Molecule - Inhibitor

Product Number
Descrizione
Specie
(+)-Pentazocine, solid,
Specie
rat, human
Amitriptyline hydrochloride, ≥98% (TLC), powder,
Specie
human
Doxepin hydrochloride, ~85% E-isomer basis, ≥98% (GC), 15% Z-isomer basis, powder,
Specie
human
Haloperidol, powder,
Specie
human, rat
Clozapine, ,
Specie
human, rat

Small Molecule - Ligand

Product Number
Descrizione
Specie
Aminobenztropine, solid,
Specie
human

Proteins

Product Number
Descrizione
Specie
ChemiScreen Membrane Preparation Human Recombinant M1 Muscarinic Acetylcholine Receptor, Human M1 GPCR membrane prepation for Radioligand binding Assays.,
Specie
human

esiRNA

Product Number
Descrizione
Specie
MISSION® esiRNA, targeting human CHRM1,
Specie
human